Design, synthesis, and anticancer evaluation of ammosamide B with pyrroloquinoline derivatives as novel BRD4 inhibitors
Wen Li, Cheng Zhang, Hong-en Zhang, Ru Dong, Jingying Liu, Chunmeng Wang, Min Wang, Yuwei Wang, Chao Wang, Yan Zhang, Lei Shi, Yong Xu, Liping Sun
Topics & Concepts
ChemistryBromodomainBRD4EpigeneticsLysineBiochemistryCancer researchStereochemistryPharmacologyGeneAmino acidBiologyProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsHistone Deacetylase Inhibitors Research