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Design, synthesis, and anticancer evaluation of ammosamide B with pyrroloquinoline derivatives as novel BRD4 inhibitors

Wen Li, Cheng Zhang, Hong-en Zhang, Ru Dong, Jingying Liu, Chunmeng Wang, Min Wang, Yuwei Wang, Chao Wang, Yan Zhang, Lei Shi, Yong Xu, Liping Sun

2022Bioorganic Chemistry10 citationsDOI

Topics & Concepts

ChemistryBromodomainBRD4EpigeneticsLysineBiochemistryCancer researchStereochemistryPharmacologyGeneAmino acidBiologyProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsHistone Deacetylase Inhibitors Research
Design, synthesis, and anticancer evaluation of ammosamide B with pyrroloquinoline derivatives as novel BRD4 inhibitors | Litcius