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Silver-mediated annulation between 5-<i>H</i>-1,2,3-thiadiazoles and 1,3-dicarbonyl compounds to construct polysubstituted furans

Mengxia Feng, Huanfeng Jiang, Liangbin Huang

2022Organic Chemistry Frontiers18 citationsDOI

Abstract

An efficient synthesis of polysubstituted furans by Ag( i )-mediated annulation between 5- H -1,2,3-thiadiazoles and 1,3-dicarbonyl compounds is reported.

Topics & Concepts

ThiadiazolesAnnulationChemistryConstruct (python library)StereochemistryCombinatorial chemistryMedicinal chemistryOrganic chemistryProgramming languageComputer scienceCatalysisCyclopropane Reaction MechanismsCatalytic C–H Functionalization MethodsCatalytic Alkyne Reactions
Silver-mediated annulation between 5-<i>H</i>-1,2,3-thiadiazoles and 1,3-dicarbonyl compounds to construct polysubstituted furans | Litcius