Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
Wenjiao Yang, Xudong Gong, Haiguo Sun, Chunhui Wu, Jin Suo, Jing Ji, Xiangrui Jiang, Jingshan Shen, He Yang, Haji Akber Aisa
Topics & Concepts
ChemistryInverse agonistAnxiolyticPartial agonistPharmacologyAgonistic behaviourAgonistIntrinsic activityRimonabantReceptorCannabinoid receptorStereochemistryPsychologyBiochemistryMedicinePsychiatryAggressionCannabis and Cannabinoid ResearchNeurotransmitter Receptor Influence on BehaviorPharmacological Receptor Mechanisms and Effects