Palladium-catalysed methylene C(sp3)–H lactamization and cycloamination enabled by chlorinated pyridine–pyridone ligands
Hau Sun Sam Chan, Yilin Lu, Jin‐Quan Yu
Topics & Concepts
ChemistryPyridineAminationPalladiumIntramolecular forceBifunctionalMedicinal chemistryMethylenePyrrolidineCombinatorial chemistryCatalysisStereochemistryOrganic chemistryCatalytic C–H Functionalization MethodsSynthesis and Catalytic ReactionsAdvanced Synthetic Organic Chemistry