Synthesis, molecular docking and enzyme inhibitory approaches of some new chalcones engrafted pyrazole as potential antialzheimer, antidiabetic and antioxidant agents
Mohammad Shahidul Islam, Abdullah Mohammed Al‐Majid, Essam Nageh Sholkamy, Sammer Yousuf, Muhammad Ayaz, Asif Nawaz, Abdul Wadood, Ashfaq Ur Rehman, Ved Prakash Verma, Ahmed Bari, Matti Haukka, Saied M. Soliman, Assem Barakat
Topics & Concepts
ChemistryChalconeDPPHPyrazoleIC50AntioxidantDocking (animal)StereochemistryNuclear chemistryBiochemistryIn vitroNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity