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RAS(ON) Therapies on the Horizon to Address KRAS Resistance: Highlight on a Phase III Clinical Candidate Daraxonrasib (RMC-6236)

Zonghui Ma, Mingxiang Zhou, Qiang Shen, Jia Zhou

2025Journal of Medicinal Chemistry12 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryKRASPhase (matter)Computational biologyCancer researchBiochemistryMutationOrganic chemistryGeneMedicineBiologyProtein Kinase Regulation and GTPase SignalingAdenosine and Purinergic SignalingRetinoids in leukemia and cellular processes
RAS(ON) Therapies on the Horizon to Address KRAS Resistance: Highlight on a Phase III Clinical Candidate Daraxonrasib (RMC-6236) | Litcius