Design, synthesis and activity study of a novel PI3K degradation by hijacking VHL E3 ubiquitin ligase
Haili Wang, Chuchu Li, Xiaoqing Liu, Ming‐Liang Ma
Topics & Concepts
Ubiquitin ligasePI3K/AKT/mTOR pathwayChemistryUbiquitinKinaseCell biologyDNA ligaseProteasomeProteolysisBiochemistryCancer researchApoptosisEnzymeBiologyGeneProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysHistone Deacetylase Inhibitors Research