Discovery of potential small molecular SARS-CoV-2 entry blockers targeting the spike protein
Lin Wang, Yan Wu, Sheng Yao, Huan Ge, Ya Zhu, Kun Chen, Wenzhang Chen, Yi Zhang, Wei Zhu, Hongyang Wang, Yu Guo, Peixiang Ma, Pengxuan Ren, Xiang-lei Zhang, Hui-qiong Li, M. Ajmal Ali, Wenqing Xu, Hualiang Jiang, Leike Zhang, Lili Zhu, Ye Yang, Weijuan Shang, Fang Bai
Topics & Concepts
Dissociation constantSurface plasmon resonanceIn silicoCoronavirusVirusSmall moleculeSpike ProteinViral entrySevere acute respiratory syndrome coronavirus 2 (SARS-CoV-2)ChemistryDrug discoveryIn vitroReceptorVirologyBiologyCoronavirus disease 2019 (COVID-19)BiochemistryViral replicationMedicineInfectious disease (medical specialty)NanotechnologyGenePathologyNanoparticleMaterials scienceDiseaseSARS-CoV-2 and COVID-19 ResearchComputational Drug Discovery MethodsCOVID-19 Clinical Research Studies