Design and synthesis of novel GluN2A NMDAR positive allosteric modulators via scaffold hopping strategy as anti-stroke therapeutic agents
Xin Chen, Hongyu Zhu, Xuequan liu, Qihong Li, Mingxin Dong
Topics & Concepts
NeuroprotectionNMDA receptorAllosteric regulationExcitotoxicityChemistryGlutamate receptorAllosteric modulatorPharmacologyIn vivoNeuroscienceReceptorBiochemistryBiologyBiotechnologyNeuroscience and Neuropharmacology ResearchMolecular Sensors and Ion DetectionIon channel regulation and function