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N-(4-acetamidophenyl)-5-acetylfuran-2-carboxamide as a novel orally available diuretic that targets urea transporters with improved PD and PK properties

Shuyuan Wang, Yue Xu, Yan Zhao, Shun Zhang, Min Li, Xiaowei Li, Jinzhao He, Hong Zhou, Zemei Ge, Runtao Li, Baoxue Yang

2021European Journal of Medicinal Chemistry16 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryBioavailabilityDiureticPharmacologyUreaIn vivoOral administrationCarboxamideBiochemistryMedicineBiologyBiotechnologyElectrolyte and hormonal disordersIon Transport and Channel RegulationAmino Acid Enzymes and Metabolism
N-(4-acetamidophenyl)-5-acetylfuran-2-carboxamide as a novel orally available diuretic that targets urea transporters with improved PD and PK properties | Litcius