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Kinase drug discovery 20 years after imatinib: progress and future directions

Philip Cohen, Darren A.E. Cross, Pasi A. Jänne

2021Nature Reviews Drug Discovery1,034 citationsDOIOpen Access PDF

Topics & Concepts

ImatinibDrug discoveryDrugMedicineImatinib mesylatePharmacologyBioinformaticsCancer researchBiologyMyeloid leukemiaChronic Myeloid Leukemia TreatmentsHER2/EGFR in Cancer ResearchPI3K/AKT/mTOR signaling in cancer
Kinase drug discovery 20 years after imatinib: progress and future directions | Litcius