Design, synthesis and biological evaluation of spiropyrazolopyridone derivatives as potent dengue virus inhibitors
Jimin Xu, Xuping Xie, Haiying Chen, Jing Zou, Yu Xue, Na Ye, Pei‐Yong Shi, Jia Zhou
Topics & Concepts
ChemistryDengue virusPotencyDengue feverTrifluoromethylStereochemistryRing (chemistry)Structure–activity relationshipChemical synthesisEC50VirusLead compoundIn vitroCombinatorial chemistryVirologyBiochemistryOrganic chemistryBiologyAlkylMosquito-borne diseases and controlResearch on Leishmaniasis StudiesViral Infections and Vectors