Design, synthesis, biological evaluation and molecular docking study of novel chalcone-based hydroxamic acids possessing a central 2, 4-dimethy pyrrole linker as potential HDAC (Histone Deacetylase) inhibitors and anticancer agents
Mozhdeh Yousefian, Maryam Hashemi, Vahid Eskandarpour, Farzin Hadizadeh, Afshin Zarghi, Razieh Ghodsi
Topics & Concepts
ChemistryChalconeVorinostatHistone deacetylaseHydroxamic acidStereochemistryDocking (animal)MTT assayHistone deacetylase inhibitorIC50HeLaCytotoxicityBiochemistryCell growthIn vitroHistoneMedicineNursingGeneHistone Deacetylase Inhibitors ResearchClick Chemistry and ApplicationsProtein Degradation and Inhibitors