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A topological switch in CFTR modulates channel activity and sensitivity to unfolding

Daniel Scholl, Maud Sigoillot, Marie Overtus, Rafael Colomer Martinez, Chloé Martens, Yiting Wang, Els Pardon, Toon Laeremans, Abel García-Pino, Jan Steyaert, David N. Sheppard, Jelle Hendrix, Cédric Govaerts

2021Nature Chemical Biology23 citationsDOIOpen Access PDF

Topics & Concepts

Cystic fibrosis transmembrane conductance regulatorCyclic nucleotide-binding domainChemistryFörster resonance energy transferBiophysicsTransmembrane domainRegulatorMutationCystic fibrosisIon channelTransmembrane proteinConformational changeMutantProtein structureCell biologyNucleotideBiochemistryBiologyGeneGeneticsFluorescenceReceptorPhysicsQuantum mechanicsCystic Fibrosis Research AdvancesAdvanced biosensing and bioanalysis techniquesNeonatal Respiratory Health Research
A topological switch in CFTR modulates channel activity and sensitivity to unfolding | Litcius