Molecular overlay-guided design of new CDK2 inhibitor thiazepinopurines: Synthesis, anticancer, and mechanistic investigations
Ebtehal M. Husseiny, Hamada S. Abulkhair, Asmaa Saleh, Najla Altwaijry, Riham A. Zidan, Fatma G. Abdulrahman
Topics & Concepts
ChemistryCyclin-dependent kinase 2Combinatorial chemistryComputational biologyNanotechnologyBiochemistryPhosphorylationProtein kinase AMaterials scienceBiologySynthesis and Reactivity of HeterocyclesClick Chemistry and Applications