Exploring biogenic chalcones as DprE1 inhibitors for antitubercular activity via in silico approach
Sanket Rathod, P.B. Chavan, Deepak Mahuli, Sneha Rochlani, Shalini Shinde, Swaranjali Pawar, Prafulla B. Choudhari, Rakesh P. Dhavale, Pralhad K. Mudalkar, Firoj A. Tamboli
Topics & Concepts
In silicoPharmacophoreMycobacterium tuberculosisTuberculosisComputational biologyQuantitative structure–activity relationshipVirtual screeningDrugChemistryDocking (animal)BiologyMedicineStereochemistryPharmacologyBiochemistryPathologyNursingGeneSynthesis and biological activityComputational Drug Discovery MethodsSynthesis and Characterization of Heterocyclic Compounds