Potency and pharmacokinetics of GS-441524 derivatives against SARS-CoV-2
Daibao Wei, Tianwen Hu, Yumin Zhang, Wei Zheng, Haitao Xue, Jingshan Shen, Yuanchao Xie, Haji Akber Aisa
Topics & Concepts
ProdrugChemistryPharmacokineticsBioavailabilityPhosphoramidatePharmacologyPotencyNucleosideMetaboliteActive metaboliteMoietyCarbamateBiochemistryStereochemistryIn vitroMedicineCOVID-19 Clinical Research StudiesSARS-CoV-2 and COVID-19 ResearchPARP inhibition in cancer therapy