On-DNA hit validation methodologies for ligands identified from DNA-encoded chemical libraries
Luca Prati, Martina Bigatti, Etienne J. Donckèle, Dario Neri, Florent Samain
Topics & Concepts
DNADNA sequencingComputational biologyLigand (biochemistry)ChemistryCombinatorial chemistryEnzymeTarget proteinBiochemistryBiologyGeneReceptorChemical Synthesis and AnalysisEnzyme function and inhibitionSynthesis and Biological Evaluation