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Selective Synthesis of Secondary Alkylboronates: Markovnikov-Selective Hydroboration of Vinylarenes with Bis(pinacolato)diboron Catalyzed by a Nickel Pincer Complex

Toru Hashimoto, Keisuke Shiota, Yoshitaka Yamaguchi

2020Organic Letters28 citationsDOI

Abstract

A nickel pincer complex bearing a β-aminoketonato-based O,N,P-tridentate ligand (1a) has been employed for the highly Markovnikov-selective hydroboration of vinylarenes using bis(pinacolato)diboron. This reaction proceeds smoothly under mild reaction conditions and affords the corresponding Markovnikov products in good to high yield.

Topics & Concepts

HydroborationChemistryMarkovnikov's rulePincer movementYield (engineering)CatalysisNickelLigand (biochemistry)Pincer ligandCombinatorial chemistryOrganic chemistryMedicinal chemistryRegioselectivityMetallurgyBiochemistryReceptorMaterials scienceOrganoboron and organosilicon chemistryCatalytic Cross-Coupling ReactionsChemical Synthesis and Analysis