Biased M1-muscarinic-receptor-mutant mice inform the design of next-generation drugs
Sophie J. Bradley, Colin Molloy, Paulina Valuskova, Louis Dwomoh, Miriam Scarpa, Mario Rossi, L. H. Finlayson, Kjell Svensson, Eyassu Chernet, Vanessa Barth, Karolina Gherbi, David A. Sykes, Caroline A. Wilson, Rajendra Mistry, Patrick M. Sexton, Arthur Christopoulos, Adrian J. Mogg, Elizabeth M. Rosethorne, Shuzo Sakata, R. A. John Challiss, Lisa M. Broad, Andrew B. Tobin
Topics & Concepts
Muscarinic acetylcholine receptorMutantMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3Computational biologyReceptorPharmacologyBiologyCell biologyChemistryMedicineGeneticsGeneReceptor Mechanisms and SignalingMonoclonal and Polyclonal Antibodies ResearchNeuropeptides and Animal Physiology