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Tripterygium wilfordii derivative celastrol, a YAP inhibitor, has antifibrotic effects in systemic sclerosis

Pratyusha Chitturi, Shiwen Xu, Bahja Ahmed Abdi, John Nguyen, David E. Carter, Sarthak Sinha, Rohit Arora, Jeff Biernaskie, Richard Stratton, Andrew Leask

2023Annals of the Rheumatic Diseases26 citationsDOI

Topics & Concepts

CelastrolFibrosisCTGFMedicineCancer researchBleomycinDermal fibroblastTransforming growth factorFibroblastPathologyBiologyGrowth factorEndocrinologyInternal medicineCell cultureApoptosisReceptorChemotherapyBiochemistryGeneticsSystemic Sclerosis and Related DiseasesHippo pathway signaling and YAP/TAZConnective Tissue Growth Factor Research
Tripterygium wilfordii derivative celastrol, a YAP inhibitor, has antifibrotic effects in systemic sclerosis | Litcius