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Design, synthesis and evaluation of oxazolopyridinone derivatives as quorum sensing inhibitors

Weijin Chen, Panpan Zhang, Ting Guo, Xiaotong Gu, Bingfang Bai, Shenyan Zhang, Xiaohong Chang, Yingmei Wang, Shutao Ma

2022Bioorganic Chemistry18 citationsDOI

Topics & Concepts

PyocyaninQuorum sensingChemistryCiprofloxacinPseudomonas aeruginosaBiofilmSwarming motilityNorfloxacinRhamnolipidMicrobiologyClarithromycinMultiple drug resistanceMinimum inhibitory concentrationAntibacterial activityIC50AntibioticsPharmacologyBacteriaBiochemistryIn vitroVirulenceBiologyGeneticsGeneBacterial biofilms and quorum sensingAntibiotic Resistance in BacteriaAntimicrobial Peptides and Activities
Design, synthesis and evaluation of oxazolopyridinone derivatives as quorum sensing inhibitors | Litcius