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Bariatric surgery reveals a gut-restricted TGR5 agonist with anti-diabetic effects

Snehal N. Chaudhari, David A. Harris, Hassan Aliakbarian, James Luo, Matthew T. Henke, Renuka Subramaniam, Ashley H. Vernon, Ali Tavakkoli, Eric G. Sheu, A. Sloan Devlin

2020Nature Chemical Biology142 citationsDOIOpen Access PDF

Topics & Concepts

G protein-coupled bile acid receptorAgonistBile acidIncretinFGF19EndogenyInternal medicineSleeve gastrectomyReceptorCholic acidGastrointestinal tractEndocrinologyGlucagon-like peptide-1HormoneExenatideChemistryType 2 diabetesMedicineDiabetes mellitusObesityWeight lossFibroblast growth factorGastric bypassDiabetes Treatment and ManagementDrug Transport and Resistance MechanismsDiet and metabolism studies
Bariatric surgery reveals a gut-restricted TGR5 agonist with anti-diabetic effects | Litcius