Discovery of novel flavonoid-based CDK9 degraders for prostate cancer treatment via a PROTAC strategy
Tizhi Wu, Zhiming Zhang, Guangyue Gong, Zekun Du, Yifan Xu, Sixian Yu, Feihai Ma, Xuan Zhang, Yuxiao Wang, Haoming Chen, Shiqi Wu, Xi Xu, Zhixia Qiu, Zhiyu Li, Hongxi Wu, Jinlei Bian, Jubo Wang, Hongxi Wu, Jinlei Bian, Jubo Wang
Topics & Concepts
FlavonoidChemistryProstate cancerPharmacologyDownregulation and upregulationCancer researchCancerBiochemistryBiologyAntioxidantGeneInternal medicineMedicineProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments