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ENT1 blockade by CNX-774 overcomes resistance to DHODH inhibition in pancreatic cancer

Nicholas J. Mullen, Ravi Thakur, Surendra K. Shukla, Nina V. Chaika, Sai Sundeep Kollala, Dezhen Wang, Chunbo He, Yuki Fujii, Shikhar Sharma, Scott E. Mulder, David B. Sykes, Pankaj K. Singh

2022Cancer Letters28 citationsDOIOpen Access PDF

Topics & Concepts

Dihydroorotate dehydrogenaseCancer researchPancreatic cancerPyrimidine metabolismKinaseBiochemistryBiologyPharmacologyChemistryPyrimidineCancerEnzymePurineGeneticsBiochemical and Molecular ResearchNeonatal Health and BiochemistryCancer, Hypoxia, and Metabolism
ENT1 blockade by CNX-774 overcomes resistance to DHODH inhibition in pancreatic cancer | Litcius