Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors
Tingting Lin, Jiacheng Li, Liping Liu, Yuan‐Qing Li, Hualiang Jiang, Kaixian Chen, Pan Xu, Cheng Luo, Bing Zhou
Topics & Concepts
Cyclin-dependent kinase 2Cyclin-dependent kinaseChemistryCyclin-dependent kinase 1Cell cultureCDK inhibitorPyrazoleKinaseCell cycleCell growthCancer researchPharmacologyApoptosisBiochemistryStereochemistryBiologyGeneticsCancer-related Molecular PathwaysAdvanced Breast Cancer TherapiesMicrotubule and mitosis dynamics