In Vitro Pharmacological Profile of KW-6356, a Novel Adenosine A2A Receptor Antagonist/Inverse Agonist
Yutaro Ohno, Michihiko Suzuki, Hidetsugu Asada, Tomoyuki Kanda, Mayumi Saki, Hikaru Miyagi, Mai Yasunaga, Chiyo Suno, So Iwata, Junichi Saito, Shinichi Uchida
Topics & Concepts
Inverse agonistAntagonismAgonistAntagonistReceptorReceptor antagonistChemistryPharmacologyCompetitive antagonistDissociation constantMedicineBiochemistryAdenosine and Purinergic SignalingReceptor Mechanisms and SignalingClick Chemistry and Applications