Rhodium-catalyzed [4+1] annulation of sulfoxonium ylides: Sequential ortho-C H functionalization/carbonyl α-amination toward polycyclic quinazolinones
Chang Wang, Peng‐Cheng Qian, Fan Chen, Jiang Cheng
Topics & Concepts
AnnulationChemistryAminationRhodiumIntramolecular forceSurface modificationArylCatalysisMedicinal chemistryRing (chemistry)Combinatorial chemistryOrganic chemistryPhysical chemistryAlkylCatalytic C–H Functionalization MethodsQuinazolinone synthesis and applicationsCancer therapeutics and mechanisms