Discovery of dihydropyridinone derivative as a covalent EZH2 degrader
Bin Zhou, Beilei Wang, Fengming Zou, Husheng Mei, Qingwang Liu, Qingwang Liu, Shuang Qi, Wenliang Wang, Rui Jin, Aoli Wang, Yongfei Chen, Feiyang Liu, Wenchao Wang, Jing Liu, Qingsong Liu, Qingsong Liu, Qingsong Liu
Topics & Concepts
EZH2ChemistryCovalent bondPRC2Drug discoveryMethylationCancer researchBiochemistryBiologyDNAOrganic chemistryEpigenetics and DNA MethylationCancer-related gene regulationRNA modifications and cancer