Litcius/Paper detail

Discovery of dihydropyridinone derivative as a covalent EZH2 degrader

Bin Zhou, Beilei Wang, Fengming Zou, Husheng Mei, Qingwang Liu, Qingwang Liu, Shuang Qi, Wenliang Wang, Rui Jin, Aoli Wang, Yongfei Chen, Feiyang Liu, Wenchao Wang, Jing Liu, Qingsong Liu, Qingsong Liu, Qingsong Liu

2023European Journal of Medicinal Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

EZH2ChemistryCovalent bondPRC2Drug discoveryMethylationCancer researchBiochemistryBiologyDNAOrganic chemistryEpigenetics and DNA MethylationCancer-related gene regulationRNA modifications and cancer