Litcius/Paper detail

Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability

Stefano Federico, Tuhina Khan, Anna Fontana, Simone Brogi, Rosaria Benedetti, Federica Sarno, Gabriele Carullo, Alex Pezzotta, A. Prasanth Saraswati, Eugenia Passaro, Luca Pozzetti, Alessandro Papa, Nicola Relitti, Sandra Gemma, Stefania Butini, Anna Pistocchi, Anna Ramunno, Fabrizio Vincenzi, Katia Varani, Vanessa Tatangelo, Laura Patrussi, Cosima T. Baldari, Simona Saponara, Beatrice Gorelli, Stefania Lamponi, Massimo Valoti, Fulvio Saccoccia, Marialaura Giannaccari, Giovina Ruberti, Daniel Herp, Manfred Jung, Lucia Altucci, Giuseppe Campiani

2022European Journal of Medicinal Chemistry29 citationsDOIOpen Access PDF

Topics & Concepts

HDAC8ChemistryHDAC6AcetylationVorinostatHistone deacetylaseBiochemistryPhenotypic screeningHistonePharmacologyCancer researchBiologyPhenotypeGeneHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and AnalysisChemical Synthesis and Analysis