Identification and validation of selective deubiquitinase inhibitors
Anthony C. Varca, Dominick Casalena, Wai Cheung Chan, Bin Hu, Robert S. Magin, Rebekka M. Roberts, Xiaoxi Liu, He Zhu, Hyuk‐Soo Seo, Sirano Dhe‐Paganon, Jarrod A. Marto, Douglas S. Auld, Sara J. Buhrlage
Topics & Concepts
Deubiquitinating enzymeUbiquitinComputational biologySmall moleculeHigh-throughput screeningFunction (biology)GeneBiologyChemistryBiochemistryGeneticsUbiquitin and proteasome pathwaysPeptidase Inhibition and AnalysisProtein Degradation and Inhibitors