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Hippo/YAP signaling’s multifaceted crosstalk in cancer

Jie Zhang, Haipeng Wu, Xinxin Ren, Zhuoshi Chen, Siyu Ye, Shuchang Chen, Jie Fang, Qirou Wu, Tiejun Zhao

2025Frontiers in Cell and Developmental Biology8 citationsDOIOpen Access PDF

Abstract

The Hippo/yes-associated protein (YAP) signaling is an evolutionarily conserved regulator in organ size control, which plays pivotal roles in cell proliferation, differentiation, apoptosis, and tissue regeneration. In cancer, dysregulation of Hippo/YAP signaling is typically recognized as one of the crucial drivers in tumorigenesis. However, beyond its canonical transcriptional targets, Hippo/YAP signaling engages in extensive crosstalk with multiple pathways to form an intricate regulatory network, thereby giving rise to its content-dependent influence on tumor initiation, progression and metastasis. This review focuses on the molecular mechanisms underlying the interplay between Hippo/YAP and pivotal signaling pathways such as nuclear factor kappa-light-chain-enhancer of activated B cells (NF-κB), wingless-type (Wnt)/β-catenin signaling pathway, transforming growth factor-beta (TGF-β), Hedgehog, Notch and other signaling pathways, as well as their implications in cancer biology. Ultimately, exploiting these mechanisms may represent promising therapeutic strategies for cancer.

Topics & Concepts

Hippo signaling pathwayCrosstalkWnt signaling pathwayBiologyCell biologySignal transductionHedgehogCarcinogenesisEnhancerNotch signaling pathwayTranscription factorCancer researchCancerGeneticsGenePhysicsOpticsHippo pathway signaling and YAP/TAZWnt/β-catenin signaling in development and cancer
Hippo/YAP signaling’s multifaceted crosstalk in cancer | Litcius