Design and synthesis of purine connected piperazine derivatives as novel inhibitors of Mycobacterium tuberculosis
Srihari Konduri, Jyothi Prashanth, Vagolu Siva Krishna, Dharmarajan Sriram, J. N. Behera, Dionicio Siegel, Koya Prabhakara Rao
Topics & Concepts
PiperazineChemistryMycobacterium tuberculosisPurineDocking (animal)StereochemistryMycobacteriumEthambutolCombinatorial chemistryBiochemistryTuberculosisEnzymeOrganic chemistryAntibioticsRifampicinNursingPathologyMedicineTuberculosis Research and EpidemiologyHIV/AIDS drug development and treatmentQuinazolinone synthesis and applications