Discovery of PHGDH inhibitors by virtual screening and preliminary structure–activity relationship study
Fu-Mao Zhang, Liang Yuan, Xin‐Wei Shi, Kai‐Rui Feng, Xiaojing Lan, Cheng Huang, Guo‐Qiang Lin, Ping Tian, Min Huang, Shuai Tang, Dingding Gao
Topics & Concepts
ChemistryEnzymeDocking (animal)NAD+ kinaseDehydrogenaseVirtual screeningBiochemistrySerineStructure–activity relationshipMutagenesisDrug discoveryIn vitroGeneMutationMedicineNursingCancer, Hypoxia, and MetabolismEpigenetics and DNA MethylationAmino Acid Enzymes and Metabolism