A multifunctional anti-AD approach: Design, synthesis, X-ray crystal structure, biological evaluation and molecular docking of chrysin derivatives
Ai‐Hong Yang, Chang Liu, Hongwei Zhang, Jianhua Wu, Rui Shen, Xiaodi Kou
Topics & Concepts
ChemistryButyrylcholinesteraseAcetylcholinesteraseDocking (animal)ChrysinStereochemistryRational designSelectivityReactive oxygen speciesChelationProton NMRCombinatorial chemistryEnzymeAchéBiochemistryOrganic chemistryAntioxidantNanotechnologyFlavonoidCatalysisMedicineMaterials scienceNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments