Dabrafenib inhibits ABCG2 and cytochrome P450 isoenzymes; potential implications for combination anticancer therapy
Aleš Šorf, Dimitrios Vagiannis, Fahda Ahmed, Jakub Hofman, Martina Čečková
Topics & Concepts
Cytochrome P450IsozymePharmacologyChemistryCYP1B1Abcg2BiochemistryMedicineEnzymeATP-binding cassette transporterTransporterGeneDrug Transport and Resistance MechanismsCancer Mechanisms and TherapyComputational Drug Discovery Methods