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Discovery of N-benzylarylamide derivatives as novel tubulin polymerization inhibitors capable of activating the Hippo pathway

Jian Song, Shenghui Wang, Chun-Hong Song, Weixin Zhang, Junxia Zhu, Xin-Yi Tian, Xiang-Jing Fu, Yan Xu, Cheng‐Yun Jin, Sai‐Yang Zhang

2022European Journal of Medicinal Chemistry29 citationsDOI

Topics & Concepts

ChemistryTubulinHippo signaling pathwayMicrotubule polymerizationMicrotubuleApoptosisCell cycleColchicineMitosisCell biologyCancer cellCell growthCell cultureBiochemistryCancerBiologyGeneticsHippo pathway signaling and YAP/TAZMicrotubule and mitosis dynamicsCell death mechanisms and regulation
Discovery of N-benzylarylamide derivatives as novel tubulin polymerization inhibitors capable of activating the Hippo pathway | Litcius