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Novel 1,2,4-triazine-quinoline hybrids: The privileged scaffolds as potent multi-target inhibitors of LPS-induced inflammatory response via dual COX-2 and 15-LOX inhibition

Amany M. Ghanim, Samar Rezq, Tarek S. Ibrahim, Damián G. Romero, Hend Kothayer

2021European Journal of Medicinal Chemistry47 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryIC50CelecoxibArachidonate 5-lipoxygenasePharmacologyIn vitroEnzymeBiochemistryArachidonic acidBiologyInflammatory mediators and NSAID effectsSynthesis and biological activitySynthesis and Biological Evaluation
Novel 1,2,4-triazine-quinoline hybrids: The privileged scaffolds as potent multi-target inhibitors of LPS-induced inflammatory response via dual COX-2 and 15-LOX inhibition | Litcius