Structure of Cytochrome P450 2C9*2 in Complex with Losartan: Insights into the Effect of Genetic Polymorphism
Sonia J. Parikh, Chiara M. Evans, Juliet O. Obi, Qinghai Zhang, Keiko Maekawa, Karen C. Glass, Manish B. Shah
Topics & Concepts
CYP2C9LosartanArginineAmino acidChemistryPolymorphism (computer science)Cytochrome P450BiochemistryAlleleBiologyGeneticsStereochemistryMetabolismAngiotensin IIReceptorGenePharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsEicosanoids and Hypertension Pharmacology