Litcius/Paper detail

Discovery of new pyrimido[5,4-c]quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies

Ramadan Ahmed Mekheimer, Samar M. R. Allam, Mariam A. Al‐Sheikh, Moustafa S. Moustafa, Saleh Mohammed Al‐Mousawi, Yaser A. Mostafa, Bahaa G. M. Youssif, Hesham A. M. Gomaa, Alaa M. Hayallah, Mohamed Abdel‐Aziz, Kamal Usef Sadek

2022Bioorganic Chemistry48 citationsDOI

Topics & Concepts

ChemistryADMECamptothecinQuinolineStereochemistryCytotoxicityIC50Docking (animal)PharmacophoreCombinatorial chemistryIn vitroBiochemistryOrganic chemistryMedicineNursingCancer therapeutics and mechanismsQuinazolinone synthesis and applicationsSynthesis and biological activity