Litcius/Paper detail

Discovery of novel 6-(piperidin-1-ylsulfonyl)-2H-chromenes targeting α-glucosidase, α-amylase, and PPAR-γ: Design, synthesis, virtual screening, and anti-diabetic activity for type 2 diabetes mellitus

Hamdy Khamees Thabet, Moustafa S. Abusaif, Mohd Imran, Mohamed H. Helal, Saleh I. Alaqel, Ahmed Alshehri, Abida Ash Mohd, Yousry A. Ammar, Ahmed Ragab

2024Computational Biology and Chemistry29 citationsDOI

Topics & Concepts

Virtual screeningType 2 Diabetes MellitusAmylasePeroxisome proliferator-activated receptorMedicineDiabetes mellitusPharmacologyChemistryComputational biologyEndocrinologyInternal medicineEnzymeDrug discoveryBiochemistryReceptorBiologyEnzyme function and inhibitionNatural Antidiabetic Agents StudiesEnzyme Catalysis and Immobilization