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Soluble Klotho Improves Hepatic Glucose and Lipid Homeostasis in Type 2 Diabetes

Huiying Gu, Wei Jiang, Nan You, Xiaobing Huang, Yuming Li, Xuehui Peng, Rui Dong, Zheng Wang, Yinan Zhu, Ke Wu, Jing Li, Lu Zheng

2020Molecular Therapy — Methods & Clinical Development70 citationsDOIOpen Access PDF

Abstract

demonstrated that sKL could inhibit the PI3K/AKT/mTORC1 signaling to upregulate peroxisome proliferator-activated receptor α (PPARα) expression by directly interacting with type 1 insulin-like growth factor receptor (IGF1R) in HFD-fed T2D mice. Thus, sKL could improve hepatic glucolipid homeostasis to ameliorate diabetic phenotypes and lipid accumulation and may function as a potential therapeutic target for the treatment of T2D and reduce the risk of NAFLD.

Topics & Concepts

EndocrinologyInternal medicineInsulin resistanceType 2 diabetesNonalcoholic fatty liver diseaseGlucose homeostasisLipid metabolismmTORC1Fatty liverInsulinDownregulation and upregulationBiologyPeroxisome proliferator-activated receptorCarbohydrate metabolismInsulin receptorSteatosisFGF21Diabetes mellitusProtein kinase BReceptorMedicineSignal transductionBiochemistryDiseaseFibroblast growth factorGeneParathyroid Disorders and TreatmentsGenetic Syndromes and ImprintingMetabolism, Diabetes, and Cancer
Soluble Klotho Improves Hepatic Glucose and Lipid Homeostasis in Type 2 Diabetes | Litcius