Design and synthesis of new quinoline-ester/-amide derivatives as potent antiproliferative agent targeting EGFR and BRAFV600E kinases
Aliaa M. Mohassab, Heba A. Hassan, Hesham A. Abou‐Zied, Mikako Fujita, Masami Otsuka, Hesham A. M. Gomaa, Bahaa G. M. Youssif, Mohamed Abdel‐Aziz
Topics & Concepts
ChemistryQuinolineDocking (animal)MoietyIC50StereochemistryEGFR inhibitorsErlotinibKinaseOximeDoxorubicinLead compoundCombinatorial chemistryIn vitroBiochemistryEpidermal growth factor receptorReceptorOrganic chemistryChemotherapyMedicineSurgeryNursingSynthesis and biological activityLung Cancer Treatments and MutationsMelanoma and MAPK Pathways