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Design, synthesis, in vitro antiproliferative evaluation and in silico studies of new VEGFR-2 inhibitors based on 4-piperazinylquinolin-2(1H)-one scaffold

Abdelfattah Hassan, Mohamed Badr, Dalia Abdelhamid, Heba A. Hassan, Mohammed A. S. Abourehab, Gamal El‐Din A. Abuo‐Rahma

2022Bioorganic Chemistry27 citationsDOI

Topics & Concepts

ChemistryStaurosporineSorafenibAngiogenesisApoptosisPharmacologyStereochemistryDocking (animal)Cell cultureKinaseCancer researchBiochemistryProtein kinase ABiologyMedicineGeneticsHepatocellular carcinomaNursingSynthesis and biological activityAngiogenesis and VEGF in CancerCancer Treatment and Pharmacology
Design, synthesis, in vitro antiproliferative evaluation and in silico studies of new VEGFR-2 inhibitors based on 4-piperazinylquinolin-2(1H)-one scaffold | Litcius