Discovery of Artesunate (ARS) PROTACs as GPX4 protein degraders for the treatment of bladder cancer
Xiyue Yang, Linghui Wang, Peiyu Lin, Yueni Ning, Yusi Lin, Yingying Xie, Congke Zhao, Lingli Mu, Cangcang Xu
Topics & Concepts
ArtesunateChemistryCancerBladder cancerPharmacologyTraditional medicineInternal medicineImmunologyMedicinePlasmodium falciparumMalariaProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis