In silico design of novel PIN1 inhibitors by combined of 3D-QSAR, molecular docking, molecular dynamic simulation and ADMET studies
Kamal Tabti, Larbi Elmchichi, Abdelouahid Sbai, Hamid Maghat, Mohammed Bouachrıne, Tahar Lakhlifi, Arabinda Ghosh
Topics & Concepts
ChemistryQuantitative structure–activity relationshipIn silicoMolecular dynamicsDocking (animal)Steric effectsMolecular modelComputational biologyStereochemistryComputational chemistryBiochemistryGeneNursingBiologyMedicineComputational Drug Discovery MethodsSynthesis and biological activityMacrophage Migration Inhibitory Factor