Synthesis and bioevaluation of novel stilbene-based derivatives as tubulin/HDAC dual-target inhibitors with potent antitumor activities in vitro and in vivo
Huajian Zhu, Wenjian Zhu, Yang Liu, Tian Gao, Jingjie Zhu, Yuchen Tan, Han Hu, Wenhao Liang, Lingyue Zhao, Jian Chen, Jian Chen, Zheying Zhu, Jichao Chen, Jichao Chen, Jinyi Xu, Shengtao Xu
Topics & Concepts
ChemistryIn vivoTubulinIn vitroApoptosisCell cultureIC50Cell cycle checkpointCell growthCell cycleCancer researchMicrotubulePharmacologyBiochemistryCell biologyBiologyBiotechnologyGeneticsHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsSynthetic Organic Chemistry Methods