Deep mutational scan of a drug efflux pump reveals its structure–function landscape
Gianmarco Meier, Sujani Thavarasah, Kai Ehrenbolger, Cedric A. J. Hutter, Lea M. Hürlimann, Jonas Barandun, Markus A. Seeger
Topics & Concepts
EffluxATP-binding cassette transporterContext (archaeology)TransporterDrugChemistryEthidium bromideP-glycoproteinBiologyBiochemistryBiophysicsMultiple drug resistancePharmacologyAntibioticsGeneDNAPaleontologyDrug Transport and Resistance MechanismsAntibiotic Resistance in BacteriaAntibiotics Pharmacokinetics and Efficacy