Diarylurea derivatives comprising 2,4-diarylpyrimidines: Discovery of novel potential anticancer agents via combined failed-ligands repurposing and molecular hybridization approaches
Ahmed Karam Farag, Ahmed H.E. Hassan, Kyung‐Sook Chung, Jeong‐Hun Lee, Hyo-Sun Gil, Kyung‐Tae Lee, Eun Joo Roh
Topics & Concepts
KinaseChemistryDrug discoveryCancer researchCancer cellPharmacologyAnnexinApoptosisCancerBiochemistryBiologyGeneticsQuinazolinone synthesis and applicationsCancer therapeutics and mechanismsSynthesis and biological activity