Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump
Nina Compagne, Juan-Carlos Jiménez-Castellanos, Virginie Meurillon, Elizabeth Pradel, Anaïs Vieira Da Cruz, Catherine Piveteau, Alexandre Biela, Maxime Eveque, Florence Leroux, Benoît Déprez, Nicolas Willand, Ruben C. Hartkoorn, Marion Flipo
Topics & Concepts
ChemistryEffluxEscherichia coliMultidrug Resistance-Associated ProteinsBiochemistryAllosteric regulationCombinatorial chemistryTransporterEnzymeATP-binding cassette transporterGeneAntibiotic Resistance in BacteriaPhenothiazines and Benzothiazines Synthesis and ActivitiesCancer therapeutics and mechanisms